Product Name

Amisulpride

CAS Number

71675-85-9

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Product Name:
Amisulpride
CAS Number:
71675-85-9
Indication:
Investigated for use/treatment in schizophrenia and schizoaffective disorders, mania in bipolar disorder, and depression.
Mode of Action:

Amisulpride binds selectively to dopamine D(2) and D(3) receptors in the limbic system. Low doses of amisulpride preferentially block presynaptic D(2)/D(3)-dopamine autoreceptors, thereby enhancing dopaminergic transmission, whereas higher doses block postsynaptic receptors, thus inhibiting dopaminergic hyperactivity. It may also have 5-ht7 antagonistic effect, useful in depression treatment.

Toxicity:

Overdoses of amisulpride have been linked with torsades de pointes.

IUPAC:
4-amino-5-(ethanesulfonyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methoxybenzamide
ATC:
N05AL05
PubChem:
2159
DrugBank:
DB06288
Formula:
C38H52N6O7
Molecular Mass:
369.479
Synonyms:
Aminosultopride
SMILES:
CCN1CCCC1CNC(=O)C1=CC(=C(N)C=C1OC)S(=O)(=O)CC
InChi:
NTJOBXMMWNYJFB-UHFFFAOYSA-N

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